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CP94253 hydrochloride

CAS No. 845861-39-4

CP94253 hydrochloride ( CP 94253 hydrochloride )

Catalog No. M27617 CAS No. 845861-39-4

CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.

Purity : >98% (HPLC)

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Datasheet

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HPLC

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Handing Instructions

Size	Price / USD	Stock	Quantity
5MG	58	Get Quote
10MG	87	Get Quote
25MG	205	Get Quote
50MG	335	Get Quote
100MG	537	Get Quote
200MG	745	Get Quote
500MG	Get Quote	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

CP94253 hydrochloride
Note

Research use only, not for human use.
Brief Description

CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
Description

CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
Synonyms

CP 94253 hydrochloride
Pathway

Others
Target

Other Targets
Recptor

panx1;Topo IV;Bacterial;DNA-gyrase
Research Area

——
Indication

——

Chemical Information

CAS Number

845861-39-4
Formula Weight

293.8
Molecular Formula

C15H20ClN3O
Purity

>98% (HPLC)
Solubility

——
SMILES

Cl.CCCOc1ccc2[nH]cc(C3=CCNCC3)c2n1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Poon IK, et al. Unexpected link between an antibiotic, pannexin channels and apoptosis. Nature. 2014 Mar 20;507(7492):329-34.

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